Opioid diketopiperazines: synthesis and activity of a prototypic class of opioid antagonists (Q44345149)

2 December 2017

title

Opioid diketopiperazines: synthesis and activity of a prototypic class of opioid antagonists (English)

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2 December 2017

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Balboni G

1

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2 December 2017

Guerrini R

2

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2 December 2017

Salvadori S

3

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Tomatis R

4

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Bryant SD

5

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Bianchi C

6

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Attila M

7

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Lazarus LH

8

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publication date

1 January 1997

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2 December 2017

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volume

378

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issue

1

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page(s)

19-29

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New and known diketopiperazines from the Caribbean sponge, Calyx cf. podatypa.

2 December 2017

cites work

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https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

The mu- and delta-opioid pharmacophore conformations of cyclic beta-casomorphin analogues indicate docking of the Phe3 residue to different domains of the opioid receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Design and synthesis of 1-aminocycloalkane-1-carboxylic acid-substituted deltorphin analogues: unique delta and mu opioid activity in modified peptides

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Preparation and opioid activity of analogues of the analgesic dipeptide 2,6-dimethyl-L-tyrosyl-N-(3-phenylpropyl)-D-alaninamide

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Molecular cloning, tissue distribution and chromosomal localization of a novel member of the opioid receptor gene family

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

21 January 2018

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https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Carnosine and related substances in animal tissues

21 January 2018

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https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Cloning of a delta opioid receptor by functional expression

21 January 2018

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https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Primary structures and expression from cDNAs of rat opioid receptor delta- and mu-subtypes.

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Identification of the amino acid residues involved in selective agonist binding in the first extracellular loop of the δ‐ and μ‐opioid receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Attempted synthesis of 2-methylalanyl-L-prolyl-L-tryptophan. An unexpected result

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Opioid receptor selectivity alteration by single residue replacement: synthesis and activity profile of [Dmt1]deltorphin B.

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Substitution on the Phe3 aromatic ring in cyclic .delta. opioid receptor-selective dermorphin/deltorphin tetrapeptide analogs: electronic and lipophilic requirements for receptor affinity

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Opioid receptor binding requirements for the delta-selective peptide deltorphin. I: Phe3 replacement with ring-substituted and heterocyclic amino acids

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Recent developments in the design of receptor specific opioid peptides

21 January 2018

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https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Effects of two diketopiperazines, cyclo (His-Pro) and Cyclo (Asp-Phe), on striatal dopamine: A microdialysis study

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

The delta-opioid receptor: isolation of a cDNA by expression cloning and pharmacological characterization

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Function of negative charge in the "address domain" of deltorphins

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Stereospecificity of amino acid side chains in deltorphin defines binding to opioid receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Interaction of deltorphin with opioid receptors: molecular determinants for affinity and selectivity

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Opioid infidelity: novel opioid peptides with dual high affinity for delta- and mu-receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

On the role of extracellular loops of opioid receptors in conferring ligand selectivity

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

The synthesis and opioid receptor binding affinities of analogues of dermorphin and its N-terminal tetrapeptide fragment with dibasic acids in position 2.

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Expression of carnosine-like immunoreactivity during retinal development in the clawed frog (Xenopus laevis).

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Role of spacer and address components in peptidomimetic .delta.-opioid receptor antagonists related to naltrindole

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Para-substituted Phe3 deltorphin analogues: enhanced selectivity of halogenated derivatives for delta opioid receptor sites

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Phe3-substituted analogues of deltorphin C. Spatial conformation and topography of the aromatic ring in peptide recognition by delta opioid receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Opioid binding profile of morphiceptin, Tyr-MIF-1 and dynorphin-related peptides in rat brain membranes

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Conformational restriction of the phenylalanine residue in a cyclic opioid peptide analog: effects on receptor selectivity and stereospecificity

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Differential stereochemical requirements of mu vs. delta opioid receptors for ligand binding and signal transduction: development of a class of potent and highly delta-selective peptide antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Conformationally restricted deltorphin analogues

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

TIPP[psi]: a highly potent and stable pseudopeptide delta opioid receptor antagonist with extraordinary delta selectivity

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Role of endogenous cyclo(His-Pro) in cold-induced hypothermia in the desert rat (Mastomys natalensis).

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Selective loss of delta opioid analgesia and binding by antisense oligodeoxynucleotides to a delta opioid receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Diketopiperazine-mediated peptide formation in aqueous solution II. Catalytic effect of phosphate

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Conversion of enkephalin and dermorphin into delta-selective opioid antagonists by single-residue substitution.

21 January 2018

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https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Selective opioid dipeptides

21 January 2018

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https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Minimum structure opioids—Dipeptide and tripeptide analogs of the enkephalins

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Amino acid composition and sequence of urinary peptides containing hydroxyproline

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Prolyl-leucyl-glycinamide, cyclo(leucylglycine), and derivatives block development of physical dependence on morphine in mice

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

Glutamate and carnosine in the vestibular system of the frog

21 January 2018

1 reference

https://api.crossref.org/works/10.1515%2FBCHM.1997.378.1.19

10.1515/BCHM.1997.378.1.19

21 January 2018

Identifiers

DOI

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2 December 2017

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