Synthesis and evaluation of derivatives of leucine enkephalin as potential affinity labels for delta opioid receptors (Q44343629)

2 December 2017

title

Synthesis and evaluation of derivatives of leucine enkephalin as potential affinity labels for delta opioid receptors (English)

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2 December 2017

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Heekyung Choi

1

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2 December 2017

Thomas F Murray

series ordinal

2

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2 December 2017

Jane V Aldrich

series ordinal

3

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2 December 2017

publication date

1 January 2003

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2 December 2017

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2 December 2017

volume

71

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2 December 2017

issue

5

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2 December 2017

page(s)

552-557

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Affinity labels for opioid receptors

2 December 2017

cites work

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6.beta.-[N,N-Bis(2-chloroethyl)amino]-17-(cyclopropylmethyl)-4,5.alpha.-epoxy-3,14-dihydroxymorphinan (chloranaltrexamine), a potent opioid receptor alkylating agent with ultralong narcotic antagonist activity

21 January 2018

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A novel opioid receptor site directed alkylating agent with irreversible narcotic antagonistic and reversible agonistic activities

21 January 2018

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Irreversible Ligands with High Selectivity Toward δ and μ Opiate Receptors

21 January 2018

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Probes for narcotic receptor mediated phenomena. 12. cis-(+)-3-Methylfentanyl isothiocyanate, a potent site-directed acylating agent for delta opioid receptors. Synthesis, absolute configuration, and receptor enantioselectivity

21 January 2018

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Naltrindole 5'-isothiocyanate: a nonequilibrium, highly selective delta opioid receptor antagonist

21 January 2018

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Reporter affinity labels: an o-phthalaldehyde derivative of beta-naltrexamine as a fluorogenic ligand for opioid receptors

21 January 2018

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Covalently induced activation of the delta opioid receptor by a fluorogenic affinity label, 7'-(phthalaldehydecarboxamido)naltrindole (PNTI).

21 January 2018

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Naphthalene dicarboxaldehyde as an electrophilic fluorogenic moiety for affinity labeling: application to opioid receptor affinity labels with greatly improved fluorogenic properties

21 January 2018

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Mutational analysis of the structure and function of opioid receptors

21 January 2018

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Highly selective photoaffinity labeling of mu and delta opioid receptors

21 January 2018

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Synthesis and biological activity of chloromethyl ketones of leucine enkephalin

21 January 2018

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Reversible affinity labeling of opioid receptors via disulfide bonding: discriminative labeling of mu and delta subtypes by chemically activated thiol-containing enkephalin analogs

21 January 2018

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Differential stereochemical requirements of mu vs. delta opioid receptors for ligand binding and signal transduction: development of a class of potent and highly delta-selective peptide antagonists

21 January 2018

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N,N-dialkylated leucine enkephalins as potential delta opioid receptor antagonists

21 January 2018

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Synthesis and evaluation of N,N-dialkyl enkephalin-based affinity labels for delta opioid receptors

21 January 2018

1 reference

Synthesis and evaluation of isothiocyanate-containing derivatives of the delta-opioid receptor antagonist Tyr-Tic-Phe-Phe (TIPP) as potential affinity labels for delta-opioid receptors

21 January 2018

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Solid phase synthesis and evaluation of Tyr-Tic-Phe-Phe(p-NHCOCH(2)Br) ([Phe(p-bromoacetamide)(4)]TIPP), a potent affinity label for delta opioid receptors

21 January 2018

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Identification of two related pentapeptides from the brain with potent opiate agonist activity

21 January 2018

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Deltakephalin, Tyr-D-Thr-Gly-Phe-Leu-Thr: a new highly potent and fully specific agonist for opiate delta-receptors

21 January 2018

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Dermorphin-based potential affinity labels for mu-opioid receptors

21 January 2018

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Synthesis and opioid activity of conformationally constrained dynorphin A analogues. 2. Conformational constraint in the "address" sequence

21 January 2018

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Comparative structure-function studies with analogs of dynorphin-(1–13) and [Leu5] enkephalin

21 January 2018

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Interaction of p-nitrophenylalanine enkephalins with mu-, delta- and kappa-subtypes of the opiate receptor.

21 January 2018

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Structure-activity relationship of biphalin. The synthesis and biological activities of new analogues with modifications in positions 3 and 4.

21 January 2018

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Synthesis of highly mu and delta opioid receptor selective peptides containing a photoaffinity group

21 January 2018

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[D-Pen2,D-Pen5]enkephalin analogues with increased affinity and selectivity for delta opioid receptors

21 January 2018

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Cyclic enkephalin analogs with exceptional potency at peripheral delta opioid receptors

21 January 2018

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Cyclic Enkephalin Analogues with Exceptional Potency and Selectivity for δ-Opioid Receptors

21 January 2018

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Substitution on the Phe3 aromatic ring in cyclic .delta. opioid receptor-selective dermorphin/deltorphin tetrapeptide analogs: electronic and lipophilic requirements for receptor affinity

21 January 2018

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Para-substituted Phe3 deltorphin analogues: enhanced selectivity of halogenated derivatives for delta opioid receptor sites

21 January 2018

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The sensitivity of opiate receptors and ligands to short wavelength ultraviolet light

21 January 2018

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Comparison of methods for the Fmoc solid-phase synthesis and cleavage of a peptide containing both tryptophan and arginine

21 January 2018

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A solid-phase synthetic strategy for the preparation of peptide-based affinity labels: synthesis of dynorphin A analogs

21 January 2018

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Synthesis and Opiate Activity in vitro of Five New p-Nitrophenylalanine4-Enkephalin-like Peptides

21 January 2018

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Para‐Substituted phenylalanine‐4 analogues of [l‐Ala3]. DPDPE: highly selective δ opioid receptor ligands

21 January 2018

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21 January 2018

Identifiers

DOI

10.1002/BIP.10533

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release_3d2j6xvhmnbznnir3kpbfarnty

2 December 2017

Fatcat ID

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Fatcat

https://api.fatcat.wiki/v0/release/3d2j6xvhmnbznnir3kpbfarnty

mapped directly with Wikidata item

24 November 2022

based on heuristic

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