2D and 3D similarity landscape analysis identifies PARP as a novel off-target for the drug Vatalanib. (Q35786901)

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24 February 2020

title

2D and 3D similarity landscape analysis identifies PARP as a novel off-target for the drug Vatalanib (English)

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24 February 2020

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ChEBI release 2020-05-28

1

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24 February 2020

Robert Preissner

7

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24 February 2020

author name string

Tim Overkamp

2

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24 February 2020

Anja Richter

3

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24 February 2020

Antje Richter

4

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24 February 2020

Peter T Daniel

5

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24 February 2020

Bernd Gillissen

6

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24 February 2020

publication date

24 September 2015

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24 February 2020

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24 February 2020

volume

16

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24 February 2020

page(s)

308

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Combination of 2D/3D ligand-based similarity search in rapid virtual screening from multimillion compound repositories. Selection and biological evaluation of potential PDE4 and PDE5 inhibitors.

24 February 2020

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Target practice: lessons from phase III trials with bevacizumab and vatalanib in the treatment of advanced colorectal cancer

12 July 2018

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Metabolism and disposition of vatalanib (PTK787/ZK-222584) in cancer patients

12 July 2018

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12 July 2018

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A FlashPlate assay for the identification of PARP-1 inhibitors

12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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12 July 2018

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25 September 2018

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21 January 2018

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21 January 2018

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12 December 2020

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Identifiers

DOI

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journals/bmcbi/GohlkeORRDGP15

24 February 2020

DBLP publication ID

1 reference

DBLP Dataset 2021-01-02

Dimensions Publication ID

28 January 2021

0 references

1 reference

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24 February 2020

PubMed publication ID

26403354

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