KUD773, a phenylthiazole derivative, displays anticancer activity in human hormone-refractory prostate cancers through inhibition of tubulin polymerization and anti-Aurora A activity. (Q35005238)

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English	KUD773, a phenylthiazole derivative, displays anticancer activity in human hormone-refractory prostate cancers through inhibition of tubulin polymerization and anti-Aurora A activity.	scientific article

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27 February 2020

KUD773, a phenylthiazole derivative, displays anticancer activity in human hormone-refractory prostate cancers through inhibition of tubulin polymerization and anti-Aurora A activity (English)

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27 February 2020

prostate cancer

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inferred from title

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27 February 2020

Konstantin Kudryavtsev

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27 February 2020

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27 February 2020

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Chia-Chun Yu

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27 February 2020

Jui-Ling Hsu

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27 February 2020

John Ta Hsu

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27 February 2020

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7 January 2015

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27 February 2020

Journal of Biomedical Science

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27 February 2020

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27 February 2020

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27 February 2020

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Creative Commons Attribution 4.0 International

7 January 2015

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April 2022 Public Data File from Crossref

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describes a project that uses

object named as

ImageQuant

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CZ Software Mentions: A large dataset of software mentions in the biomedical literature

Cytoskeleton targeting value in prostate cancer treatment

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PM060184, a new tubulin binding agent with potent antitumor activity including P-glycoprotein over-expressing tumors

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8 July 2018

2-(1H-Imidazol-1-yl)-4-[3-(trifluoro-meth-yl)phen-yl]-1,3-thia-zole.

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8 July 2018

CIL-102 induces matrix metalloproteinase-2 (MMP-2)/MMP-9 down-regulation via simultaneous suppression of genetic transcription and mRNA stability

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8 July 2018

Interaction of pseudolaric acid B with the colchicine site of tubulin

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8 July 2018

Substituted 3-(5-imidazo[2,1-b]thiazolylmethylene)-2-indolinones and analogues: synthesis, cytotoxic activity, and study of the mechanism of action

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Overexpression of active Aurora-C kinase results in cell transformation and tumour formation

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Overexpression of MMP-9 Contributes to Invasiveness of Prostate Cancer Cell Line LNCaP

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2-Phenyl-5-(pyrrolidin-1-yl)-1-(3,4,5-trimethoxybenzyl)-1H-benzimidazole, a benzimidazole derivative, inhibits growth of human prostate cancer cells by affecting tubulin and c-Jun N-terminal kinase

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8 July 2018

Aurora-a is essential for the tumorigenic capacity and chemoresistance of colorectal cancer stem cells

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8 July 2018

Synchronised phosphorylation of BNIP3, Bcl-2 and Bcl-xL in response to microtubule-active drugs is JNK-independent and requires a mitotic kinase

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8 July 2018

Beyond taxanes: a review of novel agents that target mitotic tubulin and microtubules, kinases, and kinesins.

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8 July 2018

Aurora-A kinase is essential for bipolar spindle formation and early development

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8 July 2018

Functional analysis of the Aurora Kinase A Ile31 allelic variant in human prostate

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8 July 2018

Paclitaxel: a review of adverse toxicities and novel delivery strategies.

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Chemokine and cytokine processing by matrix metalloproteinases and its effect on leukocyte migration and inflammation

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8 July 2018

Aurora kinase inhibition downregulates NF-kappaB and sensitises tumour cells to chemotherapeutic agents

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8 July 2018

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8 July 2018

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8 July 2018

Matrix metalloproteinase-7 increases resistance to Fas-mediated apoptosis and is a poor prognostic factor of patients with colorectal carcinoma

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8 July 2018

Potential antitumor agents. 37. Synthesis and antitumor activity of guanylhydrazones from imidazo[2,1-b]thiazoles and from the new heterocyclic system thiazolo[2',3':2,3]imidazo[4,5-c]quinoline

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8 July 2018

Cell death by mitotic catastrophe: a molecular definition

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8 July 2018

Overexpression and amplification of Aurora-A in hepatocellular carcinoma

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8 July 2018

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The cell cycle: a review of regulation, deregulation and therapeutic targets in cancer

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AURORA-A amplification overrides the mitotic spindle assembly checkpoint, inducing resistance to Taxol

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Aurora-B phosphorylates Histone H3 at serine28 with regard to the mitotic chromosome condensation

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26 October 2018

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10.1186/S12929-014-0107-X

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27 February 2020

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27 February 2020

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