Activity-based probes for rhomboid proteases discovered in a mass spectrometry-based assay (Q27676041)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23359682%20AND%20SRC:MED&resulttype=core&format=json

22 February 2020

title

Activity-based probes for rhomboid proteases discovered in a mass spectrometry-based assay (English)

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22 February 2020

5

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22 February 2020

Steven Verhelst

6

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22 February 2020

author name string

Oliver Vosyka

1

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22 February 2020

Kutti R Vinothkumar

2

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22 February 2020

Eliane V Wolf

3

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22 February 2020

Arwin J Brouwer

4

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22 February 2020

language of work or name

English

0 references

publication date

28 January 2013

1 reference

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Proceedings of the National Academy of Sciences of the United States of America

22 February 2020

published in

1 reference

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22 February 2020

volume

110

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22 February 2020

issue

7

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22 February 2020

page(s)

2472-2477

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Activity-based protein profiling of the Escherichia coli GlpG rhomboid protein delineates the catalytic core

22 February 2020

cites work

1 reference

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Conformational Change in Rhomboid Protease GlpG Induced by Inhibitor Binding to Its S′ Subsites

20 March 2017

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Protease signalling: the cutting edge

20 March 2017

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Insights into substrate gating in H. influenzae rhomboid

20 March 2017

1 reference

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The structural basis for catalysis and substrate specificity of a rhomboid protease

20 March 2017

1 reference

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The processing of human rhomboid intramembrane serine protease RHBDL2 is required for its proteolytic activity

20 March 2017

1 reference

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Functional and evolutionary implications of enhanced genomic analysis of rhomboid intramembrane proteases

20 March 2017

1 reference

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Open-cap conformation of intramembrane protease GlpG

20 March 2017

1 reference

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Structural basis for intramembrane proteolysis by rhomboid serine proteases

20 March 2017

1 reference

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The rhomboids: a nearly ubiquitous family of intramembrane serine proteases that probably evolved by multiple ancient horizontal gene transfers

20 March 2017

1 reference

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Reaction of porcine pancreatic elastase with 7-substituted 3-alkoxy-4-chloroisocoumarins: design of potent inhibitors using the crystal structure of the complex formed with 4-chloro-3-ethoxy-7-guanidinoisocoumarin

20 March 2017

1 reference

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Structural study of porcine pancreatic elastase complexed with 7-amino-3-(2-bromoethoxy)-4-chloroisocoumarin as a nonreactivatable doubly covalent enzyme-inhibitor complex

20 March 2017

1 reference

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Two Plasmodium rhomboid proteases preferentially cleave different adhesins implicated in all invasive stages of malaria

20 March 2017

1 reference

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Click Chemistry: Diverse Chemical Function from a Few Good Reactions

20 March 2017

1 reference

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A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

20 March 2017

1 reference

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Intramembrane proteolysis mediates shedding of a key adhesin during erythrocyte invasion by the malaria parasite

20 March 2017

1 reference

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Activity-based probes for the study of proteases: recent advances and developments.

24 May 2017

1 reference

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New approaches for dissecting protease functions to improve probe development and drug discovery

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3574917

Catalytic mechanism of rhomboid protease GlpG probed by 3,4-dichloroisocoumarin and diisopropyl fluorophosphonate

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3574917

Alkyne derivatives of isocoumarins as clickable activity-based probes for serine proteases.

29 September 2017

1 reference

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Monocyclic β-lactams are selective, mechanism-based inhibitors of rhomboid intramembrane proteases

29 September 2017

1 reference

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Current Strategies for Probing Substrate Specificity of Proteases

29 September 2017

1 reference

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Taking the plunge: integrating structural, enzymatic and computational insights into a unified model for membrane-immersed rhomboid proteolysis

29 September 2017

1 reference

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Sequence-specific intramembrane proteolysis: identification of a recognition motif in rhomboid substrates

29 September 2017

1 reference

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How intramembrane proteases bury hydrolytic reactions in the membrane.

29 September 2017

1 reference

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Intramembrane proteolysis

29 September 2017

1 reference

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Activity-based protein profiling: from enzyme chemistry to proteomic chemistry

29 September 2017

1 reference

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Rhomboid protease AarA mediates quorum-sensing in Providencia stuartii by activating TatA of the twin-arginine translocase

29 September 2017

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Structural analysis of a rhomboid family intramembrane protease reveals a gating mechanism for substrate entry

29 September 2017

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Reconstitution of intramembrane proteolysis in vitro reveals that pure rhomboid is sufficient for catalysis and specificity

29 September 2017

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Mechanism of intramembrane proteolysis investigated with purified rhomboid proteases.

29 September 2017

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Substrate specificity of rhomboid intramembrane proteases is governed by helix-breaking residues in the substrate transmembrane domain

29 September 2017

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Drosophila rhomboid-1 defines a family of putative intramembrane serine proteases

29 September 2017

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Characterization of aarA, a pleiotrophic negative regulator of the 2'-N-acetyltransferase in Providencia stuartii

29 September 2017

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Crystal structure of a rhomboid family intramembrane protease.

29 September 2017

1 reference

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Proteolytic action of GlpG, a rhomboid protease in the Escherichia coli cytoplasmic membrane

21 January 2018

1 reference

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Increased peptide deformylase activity for N-formylmethionine processing of proteins overexpressed in Escherichia coli: application to homogeneous rubredoxin production

21 January 2018

1 reference

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Activity-based protein profiling in vivo using a copper(i)-catalyzed azide-alkyne [3 + 2] cycloaddition

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.1215076110

Insights into the effect of detergents on the full-length rhomboid protease from Pseudomonas aeruginosa and its cytosolic domain

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.1215076110

Synthesis and biological evaluation of novel irreversible serine protease inhibitors using amino acid based sulfonyl fluorides as an electrophilic trap

21 January 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/23359682

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

MEROPS: the peptidase database

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/23359682

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1073/PNAS.1215076110

2 references

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23359682%20AND%20SRC:MED&resulttype=core&format=json

22 February 2020

ADS bibcode

2013PNAS..110.2472V

0 references

1 reference

2 references

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22 February 2020

PubMed publication ID

23359682

2 references

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:23359682%20AND%20SRC:MED&resulttype=core&format=json