Modulation of Androgen Receptor Activation Function 2 by Testosterone and Dihydrotestosterone (Q27646416)

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Thomas B Stanley

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Jonathan L Faggart

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Elizabeth M Wilson

Journal of Biological Chemistry

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language of work or name

English

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publication date

31 August 2007

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published in

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volume

282

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issue

35

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page(s)

25801-16

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cites work

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21 January 2018

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Androgen receptor mutations causing human androgen insensitivity syndromes show a key role of residue M807 in Helix 8-Helix 10 interactions and in receptor ligand-binding domain stability

21 January 2018

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A mechanism for androgen receptor-mediated prostate cancer recurrence after androgen deprivation therapy

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Activation Function 2 in the Human Androgen Receptor Ligand Binding Domain Mediates Interdomain Communication with the NH2-terminal Domain

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12 December 2020

Phenotypic diversity and testosterone-induced normalization of mutant L712F androgen receptor function in a kindred with androgen insensitivity

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Ligand- and coactivator-mediated transactivation function (AF2) of the androgen receptor ligand-binding domain is inhibited by the cognate hinge region

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12 December 2020

Structural basis for androgen receptor interdomain and coactivator interactions suggests a transition in nuclear receptor activation function dominance

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12 December 2020

Probing the functional link between androgen receptor coactivator and ligand-binding sites in prostate cancer and androgen insensitivity

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12 December 2020

Role of testosterone binding to the androgen receptor in male sexual differentiation of patients with 5α-reductase deficiency

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12 December 2020

A ligand-dependent bipartite nuclear targeting signal in the human androgen receptor. Requirement for the DNA-binding domain and modulation by NH2-terminal and carboxyl-terminal sequences

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Dehydroepiandrosterone activates mutant androgen receptors expressed in the androgen-dependent human prostate cancer xenograft CWR22 and LNCaP cells

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12 December 2020

Intermolecular NH2-/Carboxyl-terminal Interactions in Androgen Receptor Dimerization Revealed by Mutations That Cause Androgen Insensitivity

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12 December 2020