[18F]MK-9470, a positron emission tomography (PET) tracer for in vivo human PET brain imaging of the cannabinoid-1 receptor (Q24680848)

5

Guy Bormans

0 references

Koen Van Laere

2

Koen Van Laere

0 references

Inge De Lepeleire

15

Sandra Sanabria Bohorquez

Inge De Lepeleire

0 references

3

Sandra Sanabria-Bohórquez

0 references

Terence G Hamill

4

Terence G Hamill

0 references

Paul Rothenberg

16

Paul Rothenberg

0 references

Aubrey Stoch

17

S Aubrey Stoch

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Anne-Josée Côté

18

Josee Cote

0 references

Keith Gottesdiener

24

Keith Gottesdiener

0 references

author name string

H Donald Burns

1

0 references

Wai-si Eng

6

0 references

Ray Gibson

7

0 references

Christine Ryan

8

0 references

Brett Connolly

9

0 references

Shil Patel

10

0 references

Stephen Krause

11

0 references

Amy Vanko

12

0 references

Anne Van Hecken

13

0 references

William K Hagmann

19

0 references

James P Jewell

20

0 references

Linus S Lin

21

0 references

Ping Liu

22

0 references

Mark T Goulet

23

0 references

John A Wagner

25

0 references

Jan de Hoon

26

0 references

Luc Mortelmans

27

0 references

Tung M Fong

28

0 references

Richard J Hargreaves

Proceedings of the National Academy of Sciences of the United States of America

29

0 references

language of work or name

English

0 references

publication date

5 June 2007

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published in

0 references

volume

104

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issue

23

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page(s)

9800-5

0 references

cites work

Posterior cingulate, precuneal and retrosplenial cortices: cytology and components of the neural network correlates of consciousness

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Cannabinoid receptor localization in brain

7 April 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Identification and functional characterization of brainstem cannabinoid CB2 receptors

7 April 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

CB1 cannabinoid receptor knockout in mice leads to leanness, resistance to diet-induced obesity and enhanced leptin sensitivity

7 April 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Cannabinoids control spasticity and tremor in a multiple sclerosis model

7 April 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Kinetic modeling of N-[11C]methylpiperidin-4-yl propionate: alternatives for analysis of an irreversible positron emission tomography trace for measurement of acetylcholinesterase activity in human brain

7 April 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Characterization and localization of cannabinoid receptors in rat brain: a quantitative in vitro autoradiographic study

7 April 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Delta-9-tetrahydrocannabinol effects in schizophrenia: Implications for cognition, psychosis, and addiction

7 April 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

The PET radioligand [11C]MePPEP binds reversibly and with high specific signal to cannabinoid CB1 receptors in nonhuman primate brain

25 May 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Using positron emission tomography to facilitate CNS drug development

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Involvement of the endocannabinoid system in drug addiction

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Randomized, controlled trial of cannabis-based medicine in central pain in multiple sclerosis

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Is there a role for the endocannabinoid system in the etiology and treatment of melancholic depression?

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Imaging the dopamine system with in vivo [11C]raclopride displacement studies: understanding the true mechanism

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Endocannabinoid release from midbrain dopamine neurons: a potential substrate for cannabinoid receptor antagonist treatment of addiction.

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Endocannabinoid control of food intake and energy balance

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Prevention of Alzheimer's disease pathology by cannabinoids: neuroprotection mediated by blockade of microglial activation.

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Efficacy of two cannabis based medicinal extracts for relief of central neuropathic pain from brachial plexus avulsion: results of a randomised controlled trial

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Cannabis for dyskinesia in Parkinson disease: a randomized double-blind crossover study

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Cannabinoids and glaucoma

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

28 September 2017

Cannabis and the brain

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Cannabinoid receptors and their ligands

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Agonist-induced internalization and trafficking of cannabinoid CB1 receptors in hippocampal neurons.

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

The neurobiology of cannabinoid analgesia

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Immunohistochemical distribution of cannabinoid CB1 receptors in the rat central nervous system

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Pharmacology of cannabinoid CB1 and CB2 receptors.

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

A quantitative analysis of beta-adrenergic receptor interactions: resolution of high and low affinity states of the receptor by computer modeling of ligand binding data

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Signal sorting and amplification through G protein-coupled receptors

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Neuronal localization of cannabinoid receptors in the basal ganglia of the rat.

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Depression in Parkinson's disease is related to a genetic polymorphism of the cannabinoid receptor gene (CNR1).

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Observational analysis of feeding induced by Delta9-THC and anandamide

30 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Cannabinoid receptors in the human brain: a detailed anatomical and quantitative autoradiographic study in the fetal, neonatal and adult human brain

30 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Cannabinoid receptor binding and messenger RNA expression in human brain: an in vitro receptor autoradiography and in situ hybridization histochemistry study of normal aged and Alzheimer's brains

30 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Localization of cannabinoid receptor in the human developing and adult basal ganglia. Higher levels in the striatonigral neurons

30 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Cannabinoids reduce levodopa-induced dyskinesia in Parkinson's disease: a pilot study

30 May 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0703472104

A role for endocannabinoids in the generation of parkinsonism and levodopa-induced dyskinesia in MPTP-lesioned non-human primate models of Parkinson's disease

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0703472104

123I-labeled AM251: a radioiodinated ligand which binds in vivo to mouse brain cannabinoid CB1 receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0703472104

[123I]AM281 single-photon emission computed tomography imaging of central cannabinoid CB1 receptors before and after Delta9-tetrahydrocannabinol therapy and whole-body scanning for assessment of radiation dose in tourette patients.

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0703472104

Feasibility of central cannabinoid CB1 receptor imaging with [124I]AM281 PET demonstrated in a schizophrenic patient

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0703472104

Influence of age, postmortem delay and freezing storage period on cannabinoid receptor density and functionality in human brain.

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0703472104

Binding affinity and agonist activity of putative endogenous cannabinoids at the human neocortical CB1 receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0703472104

Characterization of CB1 cannabinoid receptor immunoreactivity in postmortem human brain homogenates.

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0703472104

An In Vitro Assay for Predicting Successful Imaging Radiotracers

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0703472104

Screening cascade and development of potential Positron Emission Tomography radiotracers for mGluR5: in vitro and in vivo characterization

21 January 2018

1 reference

https://api.crossref.org/works/10.1073%2FPNAS.0703472104

11C-JHU75528: a radiotracer for PET imaging of CB1 cannabinoid receptors

21 January 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Large receptor reserve for cannabinoid actions in the central nervous system.

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Imaging the Brain Marijuana Receptor: Development of a Radioligand that Binds to Cannabinoid CB1 Receptors In Vivo

28 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1877985

Clinical and theoretical implications of 5-HT2 and D2 receptor occupancy of clozapine, risperidone, and olanzapine in schizophrenia

28 November 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/17535893

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Internalization and Recycling of the CB1 Cannabinoid Receptor

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/17535893