Structure of the human κ-opioid receptor in complex with JDTic (Q24308048)

adenylate cyclase-inhibiting opioid receptor signaling pathway

GOA release 2020-03-11

1 reference

GOA release 2020-03-11

author

Vsevolod Katritch

4

0 references

Vadim Cherezov

15

0 references

Daniel Wacker

2

0 references

Huixian Wu

Huixian Wu

1

0 references

Xi-Ping Huang

Xi-Ping Huang

9

0 references

Bryan L. Roth

14

Bryan L Roth

0 references

Raymond C. Stevens

16

Raymond C Stevens

0 references

Gye Won Han

5

Gye Won Han

0 references

Eyal Vardy

6

Eyal Vardy

0 references

F. Ivy Carroll

10

F Ivy Carroll

0 references

Richard B Westkaemper

12

Richard B Westkaemper

0 references

Philip D Mosier

13

Philip D Mosier

0 references

Wei Liu

7

Wei Liu

0 references

author name string

Mauro Mileni

3

0 references

Aaron A Thompson

8

0 references

S Wayne Mascarella

Crystal structure of the β2 adrenergic receptor-Gs protein complex

11

0 references

language of work or name

English

0 references

publication date

17 May 2012

0 references

published in

Nature

0 references

volume

485

0 references

issue

7398

0 references

page(s)

327-32

0 references

cites work

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Analogues of (3R)-7-hydroxy-N-[(1S)-1-{[(3R,4R)-4-(3-hydroxyphenyl)-3,4-dimethyl-1-piperidinyl]methyl}-2-methylpropyl)-1,2,3,4-tetrahydro-3-isoquinolinecarboxamide (JDTic). Synthesis and in vitro and in vivo opioid receptor antagonist activity

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27 September 2017

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30 May 2018

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30 May 2018

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30 May 2018

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30 May 2018

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30 May 2018

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21 January 2018

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21 January 2018

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21 January 2018

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Human kappa opiate receptor second extracellular loop elevates dynorphin's affinity for human mu/kappa chimeras

21 January 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/22437504

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1038/NATURE10939

1 reference

Dimensions Publication ID

1053585252

0 references

Fatcat ID

release_swdaylh3ovfydictbzvosn3kwe

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/swdaylh3ovfydictbzvosn3kwe

mapped directly with Wikidata item

24 November 2022

based on heuristic

1 reference

1 reference

PubMed publication ID

22437504

1 reference