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Contents, Vol. 15, 1977

1977, Pharmacology

All rights reserved. No part of this publication may be translated into other languages, reproduced or utilized in any form or by any means, electronic or mechanical, including photo copying, recording, microcopying, or by any information storage and retrieval system, without permission in writing from the publisher.

Yol. 15, 1977 Pharmacology International Journal of Experimental and Clinical Pharmacology Editors: B.B. Brodie, Bethesda, Md. R. Domenjoz, Bonn E S. Vesetl, Hershey, Pa. Editorial Staff: H. Breuer, Bonn G.E. Gessa, Cagliari B. Holmstedt, Stockholm O. Hornykiewicz, Vienna K. Karzel, Bonn O. Kraupp, Vienna P. l.echat, Paris K. Lederis, Calgary, Alta. E.G. McQueen, Dunedin K. Mörsdorf, Bonn F. Sjöqvist, Stockholm G. Zbinden, Zurich G. Zetler, Lübeck P.A. van Zwieten, Amsterdam S. Karger • Basel • München • Paris • London • New York • Sydney All rights reserved. No part of this publication may be translated into other languages, reproduced or utilized in any form or by any means, electronic or mechanical, including photo­ copying, recording, microcopying, or by any information storage and retrieval system, without permission in writing from the publisher. © Copyright 1977 by S. Karger AG, 4011 Basel (Switzerland), Arnold-Bocklin-Strasse 25 Printed in Switzerland by Thiir AG Offsetdruck, Pratteln Contents Vol. 15, 1977 No. 1 Aceto, M.D.: Flora, R.E., and Harris, L.S.: The Effects of Naloxone and Nalorphine during the Development of Morphine Dependence in Rhesus Monkeys .............. Zimmerman, S.; Zimmerman, A.M.; Cameron, I.L., and Laurence, H.L.: A'-Tetrahydrocannabinol, Cannabidiol and Cannaliinol effects on the Immune Response of Mice ........................................................................................................................ Chaudhari, A.; Parmar, 5.5.; Singh, S.P.; Kumar, 5., and Spiro, H R.: Correlation between Antiinflammatory and Antiproteolytic Properties of Substituted Benzy lid e n e s..................................................................................................................... Anderson, G.F. and Fredericks, Ch.M.: Characterization of the Oxybutynin Antago­ nism of Drug-Induced Spasms in Detrusor ............................................................... Radd, J.P.: Marosi, J., and Fischer, J.: Comparison of the Antidiuretic Effects of Single Intravenous and Intranasal Doses of DDAVP in Diabetes insipidus ....................... Babb ini, M.; Gaiardi, M., and Bartoletti, M.: Anorexic and Behavioural Effects of a New Imidazo-Isoindole Derivative (Mazindol) in Comparison with ¿-Amphet­ amine in the Rat ....................................................................................................... Nevasaari, K.; Alakare, B., and Kdrki, N.T.: Effect of Atropine on Bile Flow and Biliary Excretion of 3H-Ouabain in the Isolated Perfused Rat Liver .................... Hine, B.; Torrelio, M., and Gershon, 5.; Analgesic, Heart Rate, and Temperature Effects of A“-THC during Acute and Chronic Administration to Conscious Rats. . Kowalewski, K. and Kokodej, A.: Effect of Secretin on Myoelectrical and Mechanical Activity of the Isolated Canine Stomach Perfused ex vivo ..................................... Adamson, R.H.; Zaharevitz, D.W., and Johns, D.G.: Enhancement of the Biological Activity of Adenosine Analogs by the Adenosine Deaminase Inhibitor 2’-Deoxycoformycin ................................................................................................................ 1 10 24 31 40 46 57 65 73 84 No. 2 Kishore, V.; Parmar, 5.5.; Kumar, 5., and Barthwal, J.P.: Anti-Inflammatory and Anti­ proteolytic Properties of Substituted Guanidines .................................................... 97 Contents IV Kun, I.; Feszt, G.; Cuparencu, B., and Orban, The Different Influence of Pre­ dominantly Antiadrenergic and Antidopaminergic Neuroleptics on the Estrous Cycle in Rats ............................................................................................................ 104 Parmar, S.S.; Chaudhary, M.; Chaudhary, S.K., and Spiro. H R.: Anticonvulsant Ac­ tivity and Selective Inhibition of NAD-Dependent Oxidations by 1,4-Disubstituted Piperazines ......................................................................................................... 112 Ercan, Z.S. and Tiirker, R.K.: Histamine Receptors in the Isolated Rat Stomach Fundus and Rabbit Aortic Strips ................................................................................118 Back. G. and Seidel, G.: Harmine Action in Rats with Lymphostatic Encephalopathy . 127 Riiegg, M. and Jaques, R.: Histamine-Releasing Effect of a Corticotrophin Derivative. I. Histamine-Releasing Effect of a Nonadecapeptide in Comparison with that of Other Histamine Liberators ........................................................................................ 134 Bodzenta, A. and Wisniewski. K.: The Effect of Prostaglandin E, on Central Cholin­ ergic Mechanisms ..........................................................................................................143 Broughton. A.C.; Secord, D.C., and Scott, G. W.: Effects of Adrenergic Stimulation on the Choledochoduodenal Sphincter M echanism ......................................................... 152 Fregly, M.J. and Rubin, M.L.: Effect of Some Substituted Pyrimidines on Develop­ ment of Desoxycorticosterone-lnduced Hypertension in R a t s .................................. 162 Haustein, K. O.: Extraordinary Cardiac Effects of 16-Epi-Gitoxin in Comparison to Ouabain in Cats and Dogs ........................................................................................... 178 No. 3 Dratman, M B.; Crutchfield, F.L.; Axelrod, J.; Utiger, R.D., and Marsh, Tri­ iodothyronine in Rat Submaxillary Salivary Gland: Effect of Altered Adrenergic Function ........................................................................................................................193 Sandor, V. and Cuparencu, B.: Analysis of the Mechanism of the Protective Activity of Some Sympathomimetic Amines in Experimental Ulcers ........................................208 Cuparencu, B. and Sandor, V.: Influence of Some Sympathomimetic Amines on the Experimental Gastric Ulcers in Rats ..........................................................................218 Turrin, M.A. and De Moraes, S.: Effects of Sammarium on the Contractile Response of the Isolated Guinea Pig Ileum to Acetylcholine, Histamine, Potassium and Barium 227 Page, J.G. and West, l..E.: Hypothermia in Rats Produced by Nabilone, a Synthetic Cannabinoid ..................................................................................................................233 Yu, J.H. and Smith, C.B.: Effect of Cocaine and Desmethylimipramine on the Uptake, Retention and Metabolism of 5H-5-Hydroxytryptamine in Rat Brain Slices . . . . 242 Severs, W.B.: Kapsha, J.M.: Klase, P.A., and Keil, L.C.: Drinking Behavior in Water Deprived Rats after Angiotensin Receptor Blockade ................................................ 254 Sirek, A.; Sirek, O.V.; Policova, Z., and Kerekes, A.: Effect of Ergot Alkaloids on Sulfonylurea-Stimulated Insulin Secretion in Dogs ...................................................259 Miller, I..; Cornett, T.: Drew, W.; McFarland, D.; Brightwell, D., and Wikler, A.: Marijuana: Dose-Response Effects on Pulse Rate, Subjective Estimates of Potency, Pleasantness, and Recognition Memory ......................................................268 Zagon, I.S. and McLaughlin. P.J.: Morphine and Brain Growth Retardation in the Rat . 276 Short Communication Datta, R.K.: Antopol, W. f. and Ghosh, J.J.: Binding of Mescaline with Subcellular Fractions upon Incubation of Brain Cortex Slices with | '"C'l Mescaline .............. 283 Contents V No. 4 Wade, A.E. and Evans, J.S.: Influence of Norethindrone on Drug-Metabolizing En­ zymes of Female Rat Liver in Various B-Vitamin Deficiency States .................... 289 Zagon, I.S. and McLaughlin, P.J.: Effects of Chronic Morphine Administration on Pregnant Rats and Their Offspring .......................................................................... 302 Belpaire, F.; Bogaert, M.; De Broe, M., and Mussche, M.; Serum Binding of Quinidine in Experimental Acute Renal F a ilu r e ....................................................................... 311 Parry, G.J.G.: Concentration of Clonazepam in Serum and Cerebrospinal Fluid of the S h e e p ............................................................................................................................. 318 Kowalewski, K. and Kolodej, A.: Effect of Intra-Arterial Infusion of Glucose on Secre­ tory Activity of Isolated Canine Stomach . ............................................................ 324 Zwieten, P.A., van: Inhibition of the Central hypotensive Effect of Clonidine by Trazodone, a Novel Antidepressant ............................................................................. 331 Smith, D.F.; Shimizu, M., and Schou, M.: Lithium Absorption, Distribution and Clearance and Body Temperature in Rats Given Lithium plus Haloperidol . . . . 337 Pham-Huu-Chanh: Pham-Huu-Chanh, A.; Clavel, P.. and Lehmann-Schad, W.: Cardio­ vascular Effects of Synthetic Substance P ...............................................................341 Kowalewski, K.: Pachkowski, T., and Secord, D.C.: Gastric Mucinous Secretion under Various Conditions of Stimulation in Hypothyroid Dogs ........................................ 348 Plowman, J.; I.akings, D.B.: Owens, E.S., and Adamson, R.H.: Initial Studies on the Penetration of Spirohydantoin Mustard into the Cerebrospinal Fluid of Dogs . . . 359 No. 5 Van Dyke, K.: Robinson, R.: Urquilla, P.: Smith, D.; Taylor, M.: Trush, M., and Wilson, M.: An Analysis of Nucleotides and Catecholamines in Bovine Medullary Granules by Anion Exchange High Pressure Liquid Chromatography and Fluorescence. Evidence that Most of the Catecholamines in Chromaffin Granules Are Stored without Associated ATP .............. . '..........................................................................377 Renis, M.; Giovine, A., and Bertolino, A.: MAO Activity in Rat Brain Stem and Cerebral Cortex following Acute and Chronic Treatment with /.-Dopa and Ethanol + L -D o p a ....................................................................................................... 392 Messiha, F.S.; Larson, J.W., and Geller, L: Voluntary Ethanol Drinking by the Rat: Effects of 2-Aminoethylisothiouronium Salt, a Modifier of NAD:NADH and Noreleagnine, a (3-Carboline Derivative ......................................................................400 Moratinos, J.; Ellis, S., and Potter, D.E.: Catecholamine-Induced Changes in Plasma Glucose and Insulin Levels in the Unanesthetized Rabbit ..................................... 407 Warwick, R.O.; Bousquet, F., and Schnell, R.C.: Effect of Acute and Chronic Morphine Treatment on Serotonin Uptake into Rat Hypothalamic Synaptosomes. 415 Severs, W.B. and Summy-Long, J. Y.: Norepinephrine-Induced Reflex Bradycardia after Central Administration of Angiotensin II ..................................................................428 Viana, A.P.: Role of Adrenergic Mechanisms in Cardiac and Respiratory Effects of Dioxin .......................................................................................................................... 436 Jaques, R.: The Pharmacological Activity of Tribenoside ................................................. 445 De Moraes, S. and Capaz, F.R.: An Analysis of the Effects of Cocaine on the Respon­ siveness of the Isolated Guinea Pig Vas deferens to Noradrenaline and Other Agonists ........................................................................................................................461 Contents VI Nousiainen, O.T.; Arnala, I.; Airaksinen, M.M., and Kokkola, K.: Potentiation of 0-Sympathomimetics with a-Adrenoceptor Blocking Drugs in Guinea Pig Trachea and Human Bronchus Preparations .......................................................................... 469 No. 6 Sirek, A.M. T.: Sirek, A., and Sirek, O. V.: Failure of Ergotamine to Alter the Lypolytic Effect of Somatotropin in D o g s ................................................................................ Fregnan, G.B. and Vidali, M.: Pharmacological Profile of a New Psychotherapeutic Agent: 4-p-Fluorophenyl-5-N(N’-o-methoxyphenyl)piperazinoethyl-4-oxazolin-2one (LR 511) ............................................................................................................. Feldman, S. and Putcha, l.: Effect of Anti-Parkinsonism Drugs on Gastric Emptying and Intestinal Transit in the Rat ................................................ ........................... Grechishkin, L.L.; Gavrovskaya, L.K., and Goldfarb, V.L.: Effect of Derivatives of 3-(0-Aminoethyl)-l ,2,4-Triazole on the Histamine H,-and H,-Receptors ............ Green, R.L.: Paradoxical Effects of Calcium-Glucagon Interaction on Cardiac Muscle Contractility of Isolated Guinea Pig Atria ....................................... ...................... Frey, H.-H.: Study into the Mechanism of Acetylsalicylic Acid-Induced Bronchoconstriction ..................................................................................................................... Mason, R. W.: The Binding of Aurothiomalate to Plasma Proteins in vitro .................... Nang, L.S.; Cosnier, D.; Terrie, G., and Moleyre.J.: Consequence of Solubility Altera­ tion by Salt Effect on Dissolution Enhancement and Biological Response of a Solid Dispersion of an Experimental Antianginal D r u g ........................................... Spierings, E.L.H.; Dzoljic, M.R., and Godschalk, M.: Effect of Clozapine on the Sleep Pattern in the R a t ....................................................................................................... Book Reviews ..................................................................... 90,191,288,367,478, Varia ...................................................... ........................................................... 288, Author In d e x ............................................................................................................... Subject Index............................................................................................................... 481 485 503 512 519 529 536 545 551 557 376 567 569