Histamine and Antihistamines

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6.

HISTAMINE AND ANTIHISTAMINES


a. Histamines
b. Antihistaminics (histamine antagonist)
b.1. H1 receptor antagonist
- Ethylene diamine: NO AVAILABLE BRANDS
b.1.1. Alkylamine
GENERIC NAME

BRAND NAME

Chlorpheniramine

ANTAMIN
CLORNAMIN
PHIL PHARMAWEALTH/ ATLANTIC
CHLORPHENAMINE

NO AVAILABLE BRANDS FOR BROMPHENIRAMINE IN THE PH


b.1.2.Piperazine
GENERIC NAME

BRAND NAME

Meclizine

BONAMINE
DIZITAB
MECLITAB

b.1.3. Phenothiazine
GENERIC NAME

BRAND NAME

Promethazine

PROMET
PROMEZIN
SYLOMET

b.2 H2 Receptor Antagonist


b.2.1. Heterocyclic Methylthioalkyl Derivative
GENERIC NAME
Cimetidine
Ranitidine

BRAND NAME
CIMULCER
TAGAMET
ACILOC
AGLOTAC
CLODINE
CONTRACID
DALYCRID
DIRANITE
ENTAC AMPOULE
LORACID
PEP-BLOC
PEPTICA
PHAREX RANITIDINE
PHIL PHARMAWEALTH/ ATLANTIC RANITIDINE
RAMADINE
RANIFIN
RANIMED

Famotidine

RANIVEX
RAXIDE
RITEMED RANITIDINE
ULCEMED
ULCEPAC
ULCERIX
ULCIN
ULZIM
ZANTAC/ ZANTAC 75
ZEPTAG
H2BLOC
HISTA-BLOC INJECTION

NO AVAILABLE BRANDS FOR NIZATIDINE IN THE PH


7. ANTIEPILEPTICS
a. Long acting barbiturates
GENERIC NAME
Phenobarbital

BRAND NAME
RHEA PHENOBARBITAL

NO AVAILABLE BRANDS FOR PRIMIDONE IN THE PH


a

Hydantoins

GENERIC NAME

Phenytoin

BRAND NAME
DILANTIN INJECTION
DILANTIN ORAL
EPILANTIN
FENEVIT
FENITIN
HOSPIRA PHENYTOIN
LANTIDIN

Succinamides
NO AVAILABLE BRANDS FOR ETHOSUXIMIDE IN THE PH

b. Dibenzazepine
GENERIC NAME

Carbamazepine

BRAND NAME
CARBAPSY
CARBASTAL
CARBAZEDIN
CARBILEPP
EPAZIN
EPIKOR
LESTROMOR
MEZACAR/MEZACAR SR
TEGREPIN
TEGRETOL

Benzodiazepine

GENERIC NAME

BRAND NAME

CLONOTRIL-0.5/CLONOTRIL-2
RIVOTRIL

Clonazepam

f.

Dialkyl acetates

GENERIC NAME

BRAND NAME
ALEPTIZ
DEPACON
DEPAKENE
DEPAMAX
EPIVAL
VALPARIN-200
VALPROS/ VALPROS i-IV

Valproic acid

g. Iminostilbenes (carbamazepine)
GENERIC NAME

BRAND NAME
CARBASTAL
CARBAPSY
CARBAZEDIN
CARBILEPP
EPAZIN
EPIKOR
LESTREMOR
MEZACAR/ MEZACAR SR
TEGREPIN
TEGRETOL

Carbamazepine

8. SEDATIVE- HYPNOTICS
a)
GENERIC NAME
Phenobarbital

Barbiturates
BRAND NAME
LUMINAL
RHEA PHENOBARBITAL

Amobarbital

N/A

Secobarbital

N/A

Thiopental

PENTAZOL
PENTHAL
PENTOBRIM
PENTOTHAL
THIOSOL

b) Benzodiazepine
GENERIC NAME
Chlordiazepoxide
Flurazepam

BRAND NAME
N/A

Triazolam
Midazolam

N/A
DORMICUM
DORMID
DORMIZOL
HYPOZAM

DALMANE

MIDAZOLEX
SEDACUM
SEDOZ
ANXIOL
ANXIONIL
NIXTENSYN
PAMIZEP
TRANKIL
VALIUM
VALZEPAM
VEXEPAM
ALTROX
AXAL
XANOR
XANOR XR
ZOLGEN
TRANXENE

Diazepam

Alprazolam
Chlorazepate

c) Piperidinediones, aldehydes and miscellaneous sedatives and hypnotics


BRAND NAME

GENERIC NAME
Gluthetimide
Chloral hydrate
Ethchlorvynol
Disulfiram
Sodium bromide

N/A
N/A
N/A
N/A
N/A
EVAZINE
ITERAX
SEDAZINE

Hydroxyzine

9. ANTIPSYCHOTICS
a.
Phenothiazine
GENERIC NAME

Chlorpromazine

Thioridazine
Prochlorpromazine
Trifluoperazine
Fluphenazine

BRAND NAME
GLOBAZINE
HARSON CHLORPROMAZINE
LARACTYL
PROMA
PROMAK
PROMAZINE
PSYNOR
THORAZINE
ZYCLORAN
MELLERIL
THIOZINE-10 / THIOZINE-25
N/A
N/A
FLUXIM
MODEZINE
SYDEPRES

b. Thioxanthenes
GENERIC NAME
Chlorprothixene
Thiothixene

BRAND NAME
N/A
N/A

c.

Butyphenones

GENERIC NAME

Haloperidol

BRAND NAME
HALDOL
HALDOL DECANOAS
SEREDOL
SEREDOL DECA
SERENACE
ZUREDEL

d. Others
GENERIC NAME
Lithium carbonate

BRAND NAME
LITCAB
MICROLIT
QUILONIUM-R

10. ANTIDEPRESSANTS
a. Hydralazine and phenylcyclopropylamines (MAP inhibitors)
GENERIC NAME
BRAND NAME
Phenelzine
N/A
b. Tricyclic Depressants
b.1 Dibenzazepine
GENERIC NAME
Desipramine
Imipramine HCl

BRAND NAME
N /A
TOFRANIL

b.2 Dibenzocycloheptadiene
GENERIC NAME
Amitryptylline

BRAND NAME
TRIPGEN

b.3 Benzotriazole Derivative


GENERIC NAME
Trazodone

BRAND NAME
N/A

12. ANALGESICS & ANTIPYRETICS


a. Opioid Analgesics, Natural Opiate & Synthetic Derivatives
a.1. Morphine
GENERIC NAME
Morphine

BRAND NAME
MORIN
MST CONTINUS

a.2. Morphine Analogues


GENERIC NAME
Codeine

BRAND NAME
N/A

Heroine
Hydromorphone
Oxycodone

N/A
N/A
OXYCONTIN
OXYNORM

a.3. Piperidines
GENERIC NAME
Meperidine
Diphenoxylate
b. Opioid Antagonist
c.
GENERIC NAME
Naloxone
Nalorphine
Lavillophan
tartrate
GENERIC NAME
Methadone
Fentanyl citrate

Pentazocine
f.

BRAND NAME
DEMEROL
N/A

BRAND NAME
NARCOTAN
NARLOX
N/A
N/A
BRAND
NAME
N/A
DUOPHARMA FENTANYL CITRATE
HOSPIRA FENTANYL CITRATE
SUBLIMAZE
TROFENTYL
N/A

Non-Addicting Analgesic and Antipyretics


d.1 Salicylates

GENERIC NAME

Acetylsalicylic Acid

BRAND NAME
ANTHROM
ASAPRIM
ASPEC-EC
ASPEN
ASPILETS/ASPILETS-EC
ASPIRIN
APITOR
ASTHROMED
BAYER ASPIRIN
BAYPRIN EC
BESPRIN

d.2 Paraaminophenol Derivatives


GENERIC NAME
Paracetamol

BRAND NAME
ACET
ACETADOL
ACF-PLUS
AEKNIL
AIZET S
ALAXAN/ALAXAN FR
ALGESIA
ALTOLAX
ALVEDON
AMACET
ANASERAN

d. Non-Opiate Addicting Analgesic


e.

Phenacetin

BAROPYRINE
BIOCET
BIOFLU
BIOGESIC
BIOPAIN
CALPOL
CLOCEPHEN
CORGIC
CORTAL FLU/CORTAL PAIN
DECOLSIN
DOLOGESIC
DOLONIL
DRINUS
DUOFLAM
FASTAMOL
FEBRILE FREE
FEBRINIL
FLEXAN
IFIMOL IV
INSOMED
KIDDILETS
LEXALGIN
MEDGENOL
MEDRACET
MULAX
MUSKELAX
MULAX
MUSKELAX
MYREMOL
NAGELIN
NAPALGIN
NAPRAN
NAPREX
NASATHERA
NORGESIC
OPIGESIC
ORNEX
OXYDOL
PANADENE
PANADOL
PARACEF
PARAGESIC
PARA-IV
PARAMED
PARVID
PYRITAS
RAPIDOL
RAXEM
RELAXID
RITEMEDPARACETAMOL
RONGESIC
SELEGERIC
SELXAN
TEMPRA
ULTRAGESIC
ZESTAGESIC
N/A

d.3 Pyrazolone
GENERIC NAME
Oxyphenbutazole
Phenylbutazone
Sulfinpyrazone

BRAND NAME
N/A
N/A
SULFIN

d.4. Agents used for treatment of gout


GENERIC
NAME

BRAND NAME
ACTIMED COLCHICINE
GOUTNIL
RHEA COLCHICINE
ALLOMARON
ALLOPRIM
ALLURASE
ALPURASE
LLANOL
LOPRIC
LORICID
PRINOL
PURINASE
SANDOZ ALLOPURINOL
TRIANOL
URINOL
ZYLOPRIM
N/A

Colchicine

Allopurinol

Probenecid
d.5.NSAIDS

d.5.1. Aryacetic acid


GENERIC NAME
Ibuprofen
Ibuprofen

Ibuprofen

Naproxen

BRAND NAME
ADVIL
ALAXAN
BRUFEN
DOLAN FP
FASPIC
FEVERFREE
FINLAX
GOFEN 400
IBUPED
MEDBUFEN
MEDBUFEN SR
MEDICOL
MEDICOL ADVANCE
FLANAX/FLANAX FORTE
NOPEN
PHAREX NAPROXEN
SKELAN

d.5.2 Indene Derivatives


GENERIC NAME
BRAND NAME
Indometacin
VI-GEL
Sulindac
N/A

GENERIC NAME
Mefenamic Acid
GENERIC
NAME
Piroxicam
Celecoxib

Diclofenac K
Diclofenac Na
Diclofenac K
Diclofenac Na
Diclofenac K

GENERIC NAME
Hydralazine

d.5.3 Fenamic Acid


BRAND NAME
ACIDAN
AFLIGEC
BRAND
NAME
ANALCID
ARTHRAN
FELDENE/FELDENE
DOLFENAL FLASH
MACROXAM TRANSDERMAL
PATCH
DOLSTEN
PALPASIN
GARDAN
ACTIMED
CELECOXIB
GISFEN
AUBREX
ISTAN
BREXEN
MEFENAX
CELCOXX
METAFLAM
250/500
CELEBREX
PHAREX
MEFENAMIC ACID
CELECURE
PONSER
CELEFLAM
PONSTAN/PONSTAN
SF
CELEXIB
RHEA MEFENAMIC
ACID
RITEMEDC-FLAM
MEFENAMIC ACID
COXBITOR
SPEGIC
FORTE
COXID
STANGENSIC
COXIDIA
SUPRAZEN/SUPRAZEN
FORTE
DANCOXIB
ZESTAN
ECOX
ACUFLAM
EUROFLAM CATAFEN
100/EUROFLAM 200
FLAMACOX
CATAFLAM
ICOX
LINCOX-100/ LINCOX-100
NACOXIB
CATAFLIN
OCCIB
PHAREXCLOFIL
CELECOXIB
PROVICOXIB
CURAFEN
RHEA CELECOXIB
SELECAP-200
DAFENAC
SWELCID
DICLON
TRUCOX
DICOFEN
VICOXIV
DICTAS
DIFENAX
MEDCLOF
MIOCLOF
NEO-PYRAZON
RHEUFLAM
RITEMED DICLOFENAC
SUBSYDE-CR
BRAND
NAME
VOLTAREN
HYLAZINE
VOTAN
HYPERZINE
PHIL PHARMAWEALTH/OBOI

a.3.Peripheral Sympatholytics
GENERIC NAME
Propranolol
Propranolol
Reserpine
Prazocin
Atenolol

BRAND NAME
INDERAL
PARVILOX
N/A
N/A
CARDIOTEN

d.5.4 others

13. CARDIOVASCULAR DRUGS


a. Antihypertensive
a.1. Diuretics
a.2.vasodilator

DURABETA
ROTELOL
TENORETIC
TENORMIN
TENORVAS
THERABLOC
TRUBLOC
ANGIMET
ANGIONORM
BETALOC
CARDIOSEL
CARDITEC
HYPETOR
METOPRIM
METOSTAD
NEOBLOC
PHAREX METOPROLOL
PROLAT/ PROLAT-DS
RITEMED METOPROLOL
BETAZOK
CARDIOSEL-OD

Metoprolol tartrate

Metoprolol
succinate

a.4. Central Alpha 2 Sympathomimetic


GENERIC NAME

BRAND NAME
CATAPIN
CATAPRES
CLONIGEN
CLONIPRESS
TERCLODINE
ALDOMET
DOPAMET
DOPARINE

Clonidine

Methylodopa

a.5. Ace Inhibitor


GENERIC NAME
Captopril
GENERIC NAME
Nifedipine

GENERIC NAME
Digoxin
Digitoxin
Enalapril
GENERIC NAME
Nitrous Acid
Amyl nitrite

BRAND NAME
BLOC-MED
BOIE CAPTOPRIL
CAPOMED
BRAND NAME
CAPTOGEN
ADALAT
HARTYLOX
NELAPINE
PHIL PHARMAWEALTH/
PANION & BF
NICARDIA/NICARDIA-XL
30
CAPTOPRIL
RITEMED CAPTOPRIL
TENSORIL
VASOSTAD
BRAND NAME
ACEBITOR
LANOXIN
CO-HYPACE
N/A
CO-RENITEC
DYNAPRIL
HYPACE
HYPRIL
NAPRILATE
BRAND
NAME
PHAREX ENALAPRIL
MALEATE
N/A
RENITEC
N/A

a.6. Calcium Channel Blocker

B. Cardiac Glycoside

c. ANTI-ANGINAL AGENTS
c.1.Nitrites

c.2.Nitrates
GENERIC NAME
Nitric Acid

BRAND NAME
N/A
DEPONIT NT 5
NITRONAL
BRAND NAME
NITROLINGUAL
INDERAL
TRANSDERM-NITRO
5
ANGIMET
ISOKET
5/10
ANGIONORM
ISOKET
RETARD 20/40
BETALOC
ISOKET
IV
BETAZOC
ISORDIL
CARDIOSEL
CARDIOSEL-OD
CARDIOSTAT
CARDITEC
HYPETOR
LOGIMAX
METOPRIM
METOSTAD
NEOBLOC
PHAREX METOPROLOL
PROLAT/PROLAT-DS
RITEMED METOPROLOL

Nitroglycerin
GENERIC NAME
Propranolol
Metoprolol
Isosorbide dinitrate

c.3.Beta blockers

c.4.Calcium antagonist
GENERIC NAME
Verapamil
Nifedipine

Diltiazem

BRAND NAME
CALAN/CALAN SR
ISOPTIN/ISOPTIN SR
SANDOZ VERAPAMIL
TARKA
BRAND NAME
ADALAT/ADALAT GITS/ADALAT RETARD
CALCIBLOC
CALCIBLOC OD
HEBLOPIN
NELAPINE
ODIPIN
ANGIOZEM
DILZEM

d. Peripheral Vasodilator
d.1. Dipiperidino
GENERIC NAME
Dypyrimidine
Dipyridamole

BRAND NAME
N/A
PERSANTIN

e. Antiarrythmic agents
e.1. Cinchona alkaloids
GENERIC NAME
Quinidine (optical isomer of quinine)

BRAND NAME
N/A

e.2. Amides
GENERIC NAME
Procainamide
Disopyramide

BRAND NAME
N/A
N/A

e.3.Xylyl derivatives
GENERIC NAME

Lidocaine

BRAND NAME
DOLOCAINE
ELIN LIDOCAINE HYDROCHLORIDE
ENDUCAINE
EURO-MED LIDOCAINE HCL
LIGNOPAD
LYGNONEX
PHIL PHARMAWEALTH / ATLANTIC LIDOCAINE
XYLOCAINE

e.4. Quaternary ammonium salts


GENERIC NAME
Bretylium

BRAND NAME
N/A

e.5. Diiodobenzyoxyethylamine
GENERIC NAME
Amiodarone

BRAND NAME
AMIO
ANOION
CORDARONE
MEDODARONE
RYTHMA

e.6. Beta-blockers
GENERIC NAME
Propanolol

Metoprolol

e.7. Ca antagonists
e.8. Hydantoins

BRAND NAME
INDERAL
ANGIMET
ANGIONORM
BETALOC
BETAZOK
CARDIOSEL
CARDIOSEL-OD
CARDIOSTAT
CARDITEC
HYPETOR
LOGIMAX
METOPRIM
METOSTAD
NEOBLOC
PHAREX METOPROLOL
PROLAT/ PROLAT-DS
RITEMED METOPROLOL

f.

Antihyperlipidemic agents
GENERIC NAME
Clofibrate
Gemfibrozil

BRAND NAME
N/A
LIPIGEM
LIPIZILE
LOPID / LOPID OD
REDUCEL

14. ANTINEOPLASTIC AGENTS


a. Alkylating agents
1. Nitrogen mustards (characterized by a bis-2-chloro-ethylamine)
GENERIC NAME
Cyclophosphamide
Chlorambucil
Melphalan

BRAND NAME
N/A
LEUKERAN
ALKERAN

2. Ethylamines
GENERIC NAME
Thiotepa

BRAND NAME
N/A

3. Alkyl sulfonates
GENERIC NAME
Busulfan

BRAND NAME
N/A

4. Nitrosoureas
GENERIC NAME
Lomustine
Carmustine
Streptozocin

BRAND NAME
N/A
N/A
N/A

5. Triazines
GENERIC NAME
Docarbazines

BRAND NAME
N/A

b. Antimetabolites
1. Folic acid antagonist
GENERIC NAME
Methotrexate

2. Purine antagonist

BRAND NAME
ALLTREX
BIOMEDIS METHOTREXATE
EMTHEXATE
HOSPIRA METHOTREXATE
MPL METHOXIL
PTERIN
TREXAN
ZEXATE

GENERIC NAME
Mercaptopurine
Thioguanine

BRAND NAME
CAPMERIN
EMPURINE
MERPURIN
PURI-NETHOL
N/A

Analogues of the natural purines


GENERIC NAME
Hypoxanthine
Guanine

BRAND NAME
N/A
N/A

3. Pyramidine antagonist
GENERIC NAME
Fluorauracil
Cytarabine

BRAND NAME
BIOMEDIS FLUOROURACIL
FIVOFLU
UTORAL
MPL CYTA
TABINE

4. Antihormone
a. Antiestrogen
GENERIC NAME

Tamoxifen citrate

b. Antiadrenal agents
c.
GENERIC NAME
Aminogluthetimide

BRAND NAME
FENAHEX
GYNATAM
GYRAXEN
MPL TAMOXIL
NOLVADEX-D
TAMOPLEX
ZITAZONIUM

BRAND NAME
N/A

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