▪ Only 6 heavy atoms were added during Hits to Leads yet the potency increased by over 6 orders o... more ▪ Only 6 heavy atoms were added during Hits to Leads yet the potency increased by over 6 orders of magnitude making this one of the most ligand efficient fragment optimisation campaigns so far described▪ Only 60 compounds were synthesis in going from fragment 1 ...
▪ Only 6 heavy atoms were added during Hits to Leads yet the potency increased by over 6 orders o... more ▪ Only 6 heavy atoms were added during Hits to Leads yet the potency increased by over 6 orders of magnitude making this one of the most ligand efficient fragment optimisation campaigns so far described▪ Only 60 compounds were synthesis in going from fragment 1 ...
Uploads
Papers by Miles Congreve